Wolverine Stack Storage & Stability Datasheet

🖨️ NovaVitality Technical Datasheet
Document ID: NV-DS-WOLV-001
Version: 1.0
Effective Date: 10 December 2025
Product: Wolverine Stack Research Blend (BPC-157 + TB-500)


⚠️ Notice: Dual-component RUO kit. Components supplied separately. No pre-mixing permitted.


1. Product Overview

ParameterSpecification
INN (Proposed)Wolverine Stack Research Blend (Protocol Name)
CAS StatusBPC-157: 137525-51-0
Molecular FormulasBPC-157: C₆₂H₉₈N₁₆O₂₂
Molecular WeightsBPC-157: 1411.55 g/mol
SequencesBPC-157: Ac-Gly-Glu-Pro-Pro-Pro-Pro-Ser-Ile-Pro-Asp-Ser-Ser-Asp-Gly-Arg-Ala-NH₂
TB-500: Ac-Ser-Asp-Lys-Pro-Asp-Met-Ala-Glu-Ile-Glu-Lys-Phe-Asp-Lys-Ser-Lys-Leu-Lys-Lys-Ser-OH
Receptor ProfileBPC-157: Integrin αvβ3/α5β1, VEGFR2
Form Supplied2× lyophilised solids (white to off-white powder) in amber glass vials
Purity (HPLC-UV)≥98% each (BPC-157: isocratic; TB-500: gradient)
Endotoxin<0.5 EU/mg each (LAL kinetic assay)
Residual SolventsMeets ICH Q3C Class 3 limits
RUO StatusFor research use only — not for human, veterinary, diagnostic, or therapeutic use
Blending StatusComponents supplied separately — pre-mixing violates MHRA GMP expectations

2. Recommended Storage Conditions

✅ Unopened (Lyophilised)

ComponentConditionStability DurationNotes
BPC-157−20°C, desiccated, dark≥36 monthsExceptionally stable (Ac/NH₂ protection)
TB-500−20°C, desiccated, dark≥24 monthsSensitive to moisture — amber vial with argon headspace
Both2–8°C≤6 monthsFor active use; log access if institutional policy requires
BothRoom Temp (≤25°C)≤7 daysTransit only — log receipt in lab register

📌 TB-500’s Met and Lys-rich domain require stricter moisture control than BPC-157.

✅ Reconstituted (Solution)

ComponentSolventShort-Term (2–8°C)Long-Term (−80°C)Notes
BPC-1570.9% NaCl≤14 days≤12 monthsHighly stable in saline
TB-5000.1% acetic acid/NaCl≤72 hours≤6 months (aliquoted)Acid suppresses aggregation
TB-500Bacteriostatic water≤48 hours≤3 monthsAcceptable; avoid neutral PBS

⚠️ Critical:
Never store mixed solutions — incompatible pH/solvents cause precipitation.
BPC-157: ≤5 freeze–thaw cycles tolerated
TB-500: ≤3 freeze–thaw cycles (aggregation risk after cycle 3)
– Use low-binding tubes for TB-500 (Lys-rich adsorbs to standard PP)


3. Stability Indicators & Degradation Risks

Risk FactorEffect on BPC-157Effect on TB-500Detection Method
MoistureMinimal (Ac/NH₂)Asp-Pro cleavage (Asp⁴–Pro⁵), Met⁶ oxidationHPLC: new peaks; LC-MS: −113 Da (Pro), +16 Da (Met)
OxidationLow (no Met/Trp/Cys)Met⁶ sulfoxide (+16 Da)LC-MS; ↓ actin binding (pyrene assay)
pH >7.0StableRapid aggregation (Lys charge neutralisation)DLS (>200 nm), visible haze
Repeated freeze–thawSlight loss (>5 cycles)Irreversible oligomerisation (>3 cycles)SEC-HPLC, reduced bioactivity
LightStableTrp¹⁴ oxidation (if present in analogues)Not applicable — native TB-500 has no Trp

🔬 Tip: For co-administration studies, prepare BPC-157 in saline (stable 14d at 4°C) and TB-500 fresh daily from −80°C stock.


4. Reconstitution Protocol (Best Practice)

For BPC-157:

  1. Equilibrate to RT (10 min).
  2. Add sterile 0.9% NaCl (e.g., 2 mL for 10 mg → 5 mg/mL).
  3. Gently swirl — dissolves in <60 sec. No filtration needed unless for in vivo.

For TB-500:

  1. Equilibrate to RT (15 min).
  2. Add 0.1% acetic acid/NaCl (e.g., 1 mL for 10 mg → 10 mg/mL).
  3. Gentle swirl → warm to 37°C (2 min) + low-power sonication (≤30 sec, ice bath).
  4. Filter through 0.22 µm PVDF.

Co-Administration Timing:
Priming protocol: BPC-157 24h pre-TB-500 (vascular/ECM priming)
Simultaneous: Inject separately (different sites) if acute model


5. Analytical Verification (Post-Storage)

TestBPC-157 AcceptanceTB-500 AcceptanceWhen to Run
HPLC Purity≥95%≥95%After >6 months storage or pre-assay
LC-MS Identity1411.5 ±1.0 Da4963.4 ±2.0 DaAnnually or after suspected degradation
Endotoxin<1.0 EU/mL<1.0 EU/mLBefore in vivo studies
Bioactivity≥90% VEGF induction (HUVECs)≥85% actin polymerisation (pyrene assay)For publication or longitudinal studies

6. References & Compliance

  • Šebečić B et al. J Physiol Pharmacol. 1996;47(2):165–172. PMID: 8877278
  • Bock SC et al. J Biol Chem. 1989;264(8):4644–4649. PMID: 2925661
  • MHRA Guidance on Unlicensed Substances in Research (Dec 2024)
  • ICH Q1A(R2): Stability Testing
  • Human Medicines Regulations 2012, Regulation 214(2) — RUO supply framework

7. Support & Documentation

📧 Technical queries: [email protected]

🔒 This datasheet is for informational purposes only. “Wolverine Stack” is a research-protocol nickname. Researchers must validate co-administration stability. NovaVitality disclaims liability for unauthorised use.